SCHEMBL9529134

SCHEMBL9529134

CCOC(=O)c1ccc(C)[n+]([O-])c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.53
CA2 P00918 4/20 0.53
CA12 O43570 3/20 0.53
CA7 P43166 3/20 0.53
CA9 Q16790 3/20 0.53
CA14 Q9ULX7 3/20 0.53
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
LMNA P02545 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAOA P21397 1/20 0.51
KMT2A Q03164 3/20 0.49
GAA P10253 1/20 0.49
CYP2C9 P11712 1/20 0.48
HPGD P15428 4/20 0.47
RECQL P46063 1/20 0.47
STS P08842 1/20 0.47
HTT P42858 2/20 0.46
MEN1 O00255 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3191323 0.83 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL30884946 0.83 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL30884942 0.83 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL30884947 0.83 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL2385010 0.82 TDP1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL30884941 0.82 KMT2A (0.49) CA1CA2CA12CA7CA9
SCHEMBL16389692 0.80 CA1 (0.46) CA1CA2CA12CA7CA9
SCHEMBL25330864 0.79 CA1 (0.45) CA1CA2CA12CA7CA9
SCHEMBL31325033 0.79 CA1 (0.45) CA1CA2CA12CA7CA9
SCHEMBL87450 0.77 CA1 (0.83) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0394476-B1 NOVEL 1,3,4-THIADIAZOLE DERIVATIVES AND ANTIULCER AGENTS CONTAINING SAME AS ACTIVE INGREDIENT TSUMURA & CO. (JP) 1993-07-28 EP disclosed
US-5106859-A CERTAIN 1,3,4-THIADIAZOLE DERIVATIVES AND ANTI-ULCER AGENT COMPRISING SAID DERIVATIVES AS ACTIVE INGREDIENT TSUMURA & CO. (JP) 1992-04-21 US disclosed
EP-0394476-A1 NOVEL 1,3,4-THIADIAZOLE DERIVATIVES AND ANTIULCER AGENTS CONTAINING SAME AS ACTIVE INGREDIENT TSUMURA & CO. (JP) 1990-10-31 EP disclosed