SCHEMBL9533759

SCHEMBL9533759

CCOC(=O)CCCN1CCC(OC(c2ccc(OC)cc2)c2ccc(OC)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 2/20 0.50
HRH1 P35367 2/20 0.50
NPC1 O15118 1/20 0.50
MLNR O43193 1/20 0.50
NR1I2 O75469 1/20 0.50
EGFR P00533 1/20 0.50
LMNA P02545 1/20 0.50
ERBB2 P04626 1/20 0.50
FYN P06241 1/20 0.50
CHRM2 P08172 1/20 0.50
CHRM4 P08173 1/20 0.50
ABCB1 P08183 1/20 0.50
ADRB1 P08588 1/20 0.50
HTR1A P08908 1/20 0.50
CHRM5 P08912 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CHRM1 P11229 1/20 0.50
ADRB3 P13945 1/20 0.50
DRD2 P14416 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9672225 0.92 BCHE (0.56) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9533482 0.91 KCNH2 (0.43) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9534850 0.88 BCHE (0.58) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL4021861 0.88 CHRM2 (0.63) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9533720 0.86 CHRM2 (0.59) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9357127 0.85 BCHE (0.60) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9531532 0.85 BCHE (0.65) HRH2HRH1NPC1MLNRNR1I2
SCHEMBL9353110 0.84 CHRM2 (0.61) HRH2HRH1NPC1MLNRNR1I2
Hydrochloric Acid SCHEMBL9353013 0.84 BCHE (0.64) HRH2HRH1NPC1MLNRNR1I2
Fumaric Acid SCHEMBL10409952 0.83 CHRM2 (0.58) HRH2HRH1NPC1MLNRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335586-B1 PIPERIDINE & PIPERAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME UBE INDUSTRIES, LTD. (JP) 1993-06-02 EP disclosed
US-4929618-A ANTIALLERGENS, ANTIHISTAMINES UBE INDUSTRIES, LTD. (JP) 1990-05-29 US disclosed
EP-0335586-A1 Piperidine & piperazine derivatives, process for preparing the same and pharmaceutical compositions containing the same UBE INDUSTRIES, LTD. (JP) 1989-10-04 EP disclosed