SCHEMBL9534253

SCHEMBL9534253

C=CCC1CCc2ccccc2C1=O

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.55
HTR1A P08908 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
ACHE P22303 1/20 0.50
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
METAP1 P53582 1/20 0.43
HTR2C P28335 1/20 0.43
CYP26A1 O43174 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9431516 0.85 CYP19A1 (0.56) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL24228697 0.84 CYP19A1 (0.57) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL874650 0.83 METAP1 (0.57) CYP19A1HTR1ASIGMAR1ACHEMETAP1
SCHEMBL11026228 0.81 CYP19A1 (0.49) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL14061976 0.79 CYP26A1 (0.64) CYP19A1ALDH1A1SMN1; SMN2TP53CYP1A2
SCHEMBL17211818 0.79 METAP1 (0.48) CYP19A1METAP1CYP26A1
SCHEMBL5608451 0.78 CYP19A1 (0.59) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL11734950 0.78 CYP19A1 (0.59) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL6307397 0.78 CYP19A1 (0.59) CYP19A1HTR1ASIGMAR1ACHEALDH1A1
SCHEMBL7305594 0.78 CYP19A1 (0.50) CYP19A1HTR1ASIGMAR1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525123-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES. UPJOHN CO (US) 1993-02-03 EP claimed
EP-0530198-A1 HETEROCYCLIC COMPOUNDS AS ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1993-03-10 EP disclosed
WO-1991015491-A1 HETEROCYCLIC COMPOUNDS AS ALDOSE REDUCTASE INHIBITORS PFIZER INC. (US) 1991-10-17 WO disclosed
US-4910212-A Containing 1,2,4-triazole or imidazole ring IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-03-20 US disclosed
EP-0281283-A1 Heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-09-07 EP disclosed