SCHEMBL9536084

SCHEMBL9536084

CCN(CCOc1cccc2c(=O)cc(N3CCOCC3)oc12)c1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 9/20 0.80
PRKDC P78527 10/20 0.60
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
PIK3CD O00329 1/20 0.53
PDE2A O00408 1/20 0.53
PIK3C2A O00443 1/20 0.53
PIK3R2 O00459 1/20 0.53
PIK3C2B O00750 1/20 0.53
BRD4 O60885 1/20 0.53
PDE5A O76074 1/20 0.53
TP53 P04637 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
PIM1 P11309 1/20 0.53
CYP2C9 P11712 1/20 0.53
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327239 0.89 P2RY12 (1.00) P2RY12
SCHEMBL7317064 0.81 PRKDC (0.68) P2RY12PRKDCKDM4EALDH1A1SMN1; SMN2
SCHEMBL910153 0.79 PRKDC (0.84) P2RY12PRKDCKDM4EALDH1A1SMN1; SMN2
SCHEMBL7328250 0.77 PRKDC (0.68) P2RY12PRKDCKDM4EALDH1A1SMN1; SMN2
SCHEMBL8799719 0.77 P2RY12 (0.79) P2RY12PRKDC
SCHEMBL8882123 0.77 P2RY12 (0.75) P2RY12PRKDCPIK3CA
SCHEMBL3542889 0.76 PRKDC (1.00) P2RY12PRKDCKDM4EALDH1A1SMN1; SMN2
SCHEMBL7326771 0.76 P2RY12 (0.82) P2RY12PRKDCKDM4EALDH1A1SMN1; SMN2
SCHEMBL9537386 0.76 P2RY12 (0.60) P2RY12PRKDC
SCHEMBL4415734 0.76 PRKDC (0.72) PRKDCKDM4EALDH1A1SMN1; SMN2PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019707-A2 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES THE UPJOHN COMPANY (US) 1991-12-26 WO claimed
EP-0525123-A1 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES. UPJOHN CO (US) 1993-02-03 EP disclosed
WO-1991019707-A2 ANTIATHEROSCLEROTIC AND ANTITHROMBOTIC 1-BENZOPYRAN-4-ONES AND 2-AMINO-1,3-BENZOXAZINE-4-ONES THE UPJOHN COMPANY (US) 1991-12-26 WO disclosed