SCHEMBL9537388

SCHEMBL9537388

C=CCC(Oc1ccccc1)C1CO1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.39
CYP2C19 P33261 1/20 0.33
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TSHR P16473 2/20 0.31
TP53 P04637 1/20 0.31
CYP3A4 P08684 1/20 0.31
HIF1A Q16665 1/20 0.31
MMP9 P14780 1/20 0.30
CHRM2 P08172 2/20 0.30
CHRM4 P08173 2/20 0.30
CHRM5 P08912 2/20 0.30
CHRM1 P11229 2/20 0.30
CHRM3 P20309 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6021886 0.78 TDP1 (0.42) TDP1ALDH1A1SMN1; SMN2TSHRTP53
SCHEMBL28675474 0.75 TDP1 (0.40) TDP1ALDH1A1SMN1; SMN2TSHRTP53
SCHEMBL20388803 0.75 TDP1 (0.40) TDP1CHRM2CHRM4CHRM5CHRM1
SCHEMBL9589101 0.75 MEN1 (0.37) TDP1ALDH1A1
SCHEMBL671115 0.75 TDP1 (0.38) TDP1TSHRCHRM2CHRM4CHRM5
SCHEMBL9132176 0.73 CYP3A4 (0.44) CYP2C19ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL3402458 0.73 TDP1 (0.35) TDP1ALDH1A1
SCHEMBL9132179 0.72 CYP3A4 (0.40) TDP1CYP2C19ALDH1A1KDM4EMAPT
SCHEMBL27259892 0.71 CYP2C19 (0.43) CYP2C19ALDH1A1KDM4EMAPTALOX15
SCHEMBL1778182 0.71 CYP2C19 (0.41) CYP2C19ALDH1A1KDM4EMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed