SCHEMBL9538527

SCHEMBL9538527

OC(CNC1CCc2ccccc2C1)COc1ccccc1Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.72
CYP1A2 P05177 2/20 0.72
CYP3A4 P08684 2/20 0.72
TSHR P16473 2/20 0.72
CYP2C19 P33261 2/20 0.72
CYP2D6 P10635 1/20 0.72
CYP2C9 P11712 1/20 0.72
THPO P40225 1/20 0.72
NPC1 O15118 1/20 0.72
MTOR P42345 1/20 0.72
RAB9A P51151 1/20 0.72
KMT2A Q03164 7/20 0.67
MEN1 O00255 5/20 0.67
KDM4E B2RXH2 2/20 0.67
LMNA P02545 2/20 0.67
GMNN O75496 1/20 0.67
PMP22 Q01453 1/20 0.67
NPY1R P25929 1/20 0.59
PRMT5 O14744 2/20 0.54
ADRB1 P08588 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534612 0.90 TP53 (0.60) TP53CYP1A2CYP3A4TSHRCYP2C19
Hydrochloric Acid SCHEMBL9587219 0.89 TP53 (0.59) TP53CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL9535328 0.86 CYP1A2 (0.76) TP53CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL9537748 0.86 CYP1A2 (0.76) TP53CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL9536180 0.85 TP53 (0.69) TP53CYP1A2CYP3A4TSHRCYP2C19
Hydrochloric Acid SCHEMBL9589088 0.85 CYP1A2 (0.74) TP53CYP1A2CYP3A4TSHRCYP2C19
Hydrochloric Acid SCHEMBL9587965 0.85 CYP1A2 (0.74) TP53CYP1A2CYP3A4TSHRCYP2C19
Hydrochloric Acid SCHEMBL9588401 0.84 TP53 (0.67) TP53CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL9537913 0.84 CYP1A2 (0.70) TP53CYP1A2CYP3A4TSHRCYP2C19
SCHEMBL9536903 0.84 NPY1R (0.84) TP53CYP1A2CYP3A4TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5254595-A Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them ELF SANOFI (FR) 1993-10-19 US disclosed
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed
EP-0375560-A1 Aryloxypropanolaminotetralines, process for their preparation and pharmaceutical compositions containing same ELF SANOFI (FR) 1990-06-27 EP disclosed