SCHEMBL9539636

SCHEMBL9539636

COc1cc(CCl)c(O)c2c1C(=O)c1ccccc1C2=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.67
AURKB Q96GD4 1/20 0.67
MAPT P10636 5/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 3/20 0.54
TDP1 Q9NUW8 3/20 0.54
USP2 O75604 1/20 0.54
DUSP3 P51452 1/20 0.54
RAB9A P51151 4/20 0.52
NPC1 O15118 2/20 0.52
SMN1; SMN2 Q16637 3/20 0.47
MAPK1 P28482 2/20 0.47
POLB P06746 2/20 0.47
FGB P02675 1/20 0.47
THRB P10828 1/20 0.47
ADORA2A P29274 1/20 0.47
PPARG P37231 1/20 0.47
NCOA2 Q15596 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9539660 0.84 MAPT (0.53) AURKAAURKBMAPTMEN1KMT2A
SCHEMBL23043842 0.82 MAPT (0.66) MAPTMEN1KMT2AALDH1A1KDM4E
SCHEMBL12581679 0.80 MAPT (0.64) MAPTMEN1KMT2AALDH1A1KDM4E
SCHEMBL28727751 0.80 AURKA (1.00) AURKAAURKBMAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL9539622 0.80 AURKA (0.55) AURKAAURKBALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL9539442 0.79 AURKA (0.54) AURKAAURKBALDH1A1KDM4ESMN1; SMN2
SCHEMBL19341713 0.79 MAPT (0.61) MAPTMEN1KMT2AALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9538671 0.76 AURKA (0.51) AURKAAURKBMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL9539440 0.76 AURKA (0.50) AURKAAURKBMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL9542152 0.73 KDM4E (0.50) AURKAAURKBMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993005054-A1 OXAZAPHOSPHORINES USEFUL AS ANTITUMOR AGENTS, A PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-03-18 WO disclosed