SCHEMBL9539804

SCHEMBL9539804

CCC(N)C(=O)c1cccc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.53
SLC6A2 P23975 5/20 0.51
SLC6A3 Q01959 4/20 0.51
CHRNA1 P02708 2/20 0.51
CHRNG P07510 2/20 0.51
CHRNB1 P11230 2/20 0.51
CHRNB2 P17787 2/20 0.51
CHRNB4 P30926 2/20 0.51
SLC6A4 P31645 2/20 0.51
CHRNA3 P32297 2/20 0.51
CHRNA4 P43681 2/20 0.51
CHRND Q07001 2/20 0.51
ITGA5 P08648 1/20 0.51
CYP2C19 P33261 1/20 0.51
HRH1 P35367 1/20 0.51
CHRNA7 P36544 1/20 0.51
OPRK1 P41145 1/20 0.51
KCNH2 Q12809 1/20 0.51
ALDH1A1 P00352 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1093383 0.81 SLC6A2 (0.56) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL15007460 0.81 SLC6A2 (0.53) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL20809637 0.81 SLC6A2 (0.56) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL2599163 0.81 SLC6A2 (0.53) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL9559781 0.81 PARP1 (0.55) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL3851904 0.81 SLC6A2 (0.59) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL3852863 0.81 SLC6A2 (0.59) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL9041221 0.81 SLC6A2 (0.59) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL633919 0.80 SLC6A2 (0.51) PARP1SLC6A2SLC6A3CHRNA1CHRNG
SCHEMBL2290370 0.80 SLC6A2 (0.51) PARP1SLC6A2SLC6A3CHRNA1CHRNG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed