SCHEMBL9540129

SCHEMBL9540129

CCCC1(C2CC2)c2cc(Cl)ccc2N(Cc2ccc(OC)cc2)C(=O)N1CC1CC1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.43
OPRL1 P41146 13/20 0.41
OPRM1 P35372 12/20 0.40
SCN9A Q15858 1/20 0.39
CMA1 P23946 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540045 0.92 PTGDR2 (0.45) PTGDR2OPRL1OPRM1SCN9ACMA1
SCHEMBL9542817 0.87 PTGDR2 (0.47) PTGDR2OPRL1SCN9ACMA1
SCHEMBL9539893 0.83 PTGDR2 (0.42) PTGDR2OPRL1OPRM1SCN9ACMA1
SCHEMBL9539749 0.83 PTGDR2 (0.43) PTGDR2OPRL1OPRM1SCN9ACMA1
SCHEMBL9541585 0.83 PTGDR2 (0.45) PTGDR2OPRL1SCN9ACMA1
SCHEMBL9540141 0.83 PTGDR2 (0.47) PTGDR2OPRL1OPRM1SCN9ACMA1
SCHEMBL9540043 0.81 PTGDR2 (0.47) PTGDR2OPRL1SCN9ACMA1
SCHEMBL9541633 0.80 PTGDR2 (0.44) PTGDR2OPRL1OPRM1SCN9ACMA1
SCHEMBL9541601 0.79 PTGDR2 (0.47) PTGDR2OPRL1SCN9ACMA1
SCHEMBL9539017 0.79 PTGDR2 (0.49) PTGDR2SCN9ACMA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed