SCHEMBL9540137

SCHEMBL9540137

C=CCC1(C2CC2)NC(=O)N(Cc2ccc(OC)cc2)c2ccc(Cl)cc21

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 8/20 0.47
SCN9A Q15858 2/20 0.41
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
CMA1 P23946 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
TP53 P04637 1/20 0.38
BLM P54132 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
OPRL1 P41146 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539935 0.89 PTGDR2 (0.44) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9540078 0.87 PTGDR2 (0.49) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9540101 0.86 PTGDR2 (0.46) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9539009 0.86 PTGDR2 (0.46) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9540160 0.86 PTGDR2 (0.46) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9542778 0.85 PTGDR2 (0.47) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9539054 0.85 PTGDR2 (0.48) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9539778 0.85 PTGDR2 (0.45) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9539122 0.84 PTGDR2 (0.45) PTGDR2SCN9AMEN1ALDH1A1MAPT
SCHEMBL9539940 0.84 PTGDR2 (0.43) PTGDR2SCN9AMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed