SCHEMBL9540142

SCHEMBL9540142

O=C1Nc2ccc(Cl)cc2C(COc2ccccc2)(C2CC2)N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 3/20 0.44
AKR1B1 P15121 5/20 0.37
ADAMTS5 Q9UNA0 4/20 0.37
ADAMTS4 O75173 2/20 0.37
MMP13 P45452 2/20 0.37
MMP2 P08253 1/20 0.37
ADAMTS1 Q9UHI8 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
AKR1A1 P14550 2/20 0.36
MAOB P27338 1/20 0.35
CBX7 O95931 1/20 0.35
CDYL Q9Y232 1/20 0.35
ADAM17 P78536 2/20 0.35
ELOVL6 Q9H5J4 1/20 0.35
MMP1 P03956 1/20 0.35
MMP12 P39900 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541537 0.81 PDE7A (0.46) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9539045 0.78 PDE7A (0.50) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9539196 0.77 PDE7A (0.49) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9571241 0.77 PDE7A (0.49) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9539773 0.76 PDE7A (0.48) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9539898 0.75 PDE7A (0.47) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9539949 0.75 PDE7A (0.47) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9542754 0.74 PDE7A (0.46) PDE7AAKR1B1ADAMTS5ADAMTS4MMP13
SCHEMBL9541586 0.73 PTGDR2 (0.45)
SCHEMBL9571188 0.71 PDE7A (0.45) PDE7AAKR1B1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed