SCHEMBL9541153

SCHEMBL9541153

CNCC[C@@H]1CCN(c2c(F)c(N)c3c(=O)c(C(=O)O)cn(C4CC4)c3c2OC)C1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.58
GSK3B P49841 12/20 0.55
POLB P06746 2/20 0.53
CACNA1F O60840 1/20 0.53
MAPK1 P28482 1/20 0.53
CACNA1D Q01668 1/20 0.53
CACNA1S Q13698 1/20 0.53
CACNA1C Q13936 1/20 0.53
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
PRKD3 O94806 1/20 0.47
ALOX15 P16050 1/20 0.47
OPRM1 P35372 1/20 0.47
CLK2 P49760 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688856 0.92 KCNH2 (0.59) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9428498 0.92 KCNH2 (0.63) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9428507 0.92 KCNH2 (0.63) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9457226 0.91 KCNH2 (0.65) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9457828 0.91 KCNH2 (0.65) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9457229 0.91 KCNH2 (0.65) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL10698651 0.89 POLB (0.55) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9688237 0.88 KCNH2 (0.59) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9688853 0.87 KCNH2 (0.59) KCNH2GSK3BPOLBCACNA1FMAPK1
SCHEMBL9372691 0.85 KCNH2 (0.60) KCNH2GSK3BPOLBCACNA1FMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559774-A1 INDIVIDUAL STEREOISOMERS OF 7- 3-(1-AMINOALKYL)-1-PYRROLIDINYL]-QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1993-09-15 EP claimed