SCHEMBL9541570

SCHEMBL9541570

O=C1Nc2ccc(Cl)cc2C(CCO)(CC2CC2)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 2/20 0.46
AKR1B1 P15121 4/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
IDO1 P14902 2/20 0.37
AKR1A1 P14550 1/20 0.35
ELOVL6 Q9H5J4 1/20 0.34
CYP46A1 Q9Y6A2 2/20 0.34
MMP2 P08253 1/20 0.33
ADAMTS5 Q9UNA0 1/20 0.33
NR1I2 O75469 1/20 0.33
NR3C1 P04150 1/20 0.33
PGR P06401 1/20 0.33
ADRB1 P08588 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
MAPT P10636 1/20 0.33
CNR1 P21554 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540113 0.90 PDE7A (0.52) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9539947 0.82 PDE7A (0.45) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9571241 0.79 PDE7A (0.49) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9539045 0.77 PDE7A (0.50) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9538943 0.74 PDE7A (0.47) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9539149 0.70 PTGDR2 (0.45) MEN1KMT2AMAPT
SCHEMBL9540154 0.70 PDE7A (0.50) PDE7AAKR1B1IDO1AKR1A1PGR
SCHEMBL9539063 0.69 AKR1B1 (0.47) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9539196 0.68 PDE7A (0.49) PDE7AAKR1B1MEN1KMT2AIDO1
SCHEMBL9539072 0.67 PDE7A (0.57) PDE7AAKR1B1MEN1KMT2AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed