SCHEMBL9541577

SCHEMBL9541577

O=c1nc2ccc(Cl)cc2c(-c2ccccc2)n1C1CCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
LMNA P02545 2/20 0.45
HTT P42858 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
FABP4 P15090 2/20 0.43
FABP5 Q01469 2/20 0.43
GAA P10253 1/20 0.42
ALOX15 P16050 1/20 0.42
MAT2A P31153 1/20 0.42
EGFR P00533 1/20 0.41
FABP3 P05413 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
MEN1 O00255 1/20 0.40
ATM Q13315 1/20 0.40
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
DHODH Q02127 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540165 0.95 KDM4E (0.47) KDM4ELMNAHTTL3MBTL1FABP4
SCHEMBL9540062 0.76 KDM4E (0.51) KDM4ELMNAHTTL3MBTL1FABP4
SCHEMBL11635515 0.76 MAPT (0.47) KDM4ELMNAHTTGAAALOX15
SCHEMBL9540153 0.73 KDM4E (0.50) KDM4ELMNAHTTL3MBTL1FABP4
SCHEMBL9539113 0.73 KDM4E (0.48) KDM4ELMNAHTTL3MBTL1FABP4
SCHEMBL9542746 0.69 HRH3 (0.42) MAT2AKCNH2HRH3NPC1RAB9A
SCHEMBL25373437 0.68 MAPK8 (0.51) FABP4FABP5
SCHEMBL9539742 0.66 AURKA (0.52) KDM4ELMNAHTTL3MBTL1EGFR
SCHEMBL25373040 0.65 MAPK8 (0.51) FABP4FABP5
SCHEMBL9539747 0.65 KDM4E (0.47) KDM4ELMNAHTTL3MBTL1FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530994-A1 Quinazoline derivatives as inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1993-03-10 EP disclosed
WO-1993004047-A1 QUINAZOLINE DERIVATIVES AS INHIBITORS OF HIV REVERSE TRANSCRIPTASE MERCK & CO., INC. (US) 1993-03-04 WO disclosed