SCHEMBL9552802

SCHEMBL9552802

N#CCCCCc1ccc(-c2ccc(CCC#N)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HIF1A Q16665 2/20 0.38
EPAS1 Q99814 2/20 0.38
RARB P10826 5/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
ALDH1A1 P00352 1/20 0.36
RARA P10276 1/20 0.36
MAPT P10636 1/20 0.36
MTOR P42345 1/20 0.36
HDAC2 Q92769 1/20 0.35
FDFT1 P37268 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9553703 0.96 TSHR (0.52) TSHRHSD17B10MEN1KMT2AHIF1A
SCHEMBL9553062 0.96 TSHR (0.52) TSHRHSD17B10MEN1KMT2AHIF1A
SCHEMBL9552742 0.89 TSHR (0.48) TSHRHSD17B10MEN1KMT2ARARB
SCHEMBL9553570 0.89 TSHR (0.48) TSHRHSD17B10MEN1KMT2ARARB
SCHEMBL9552869 0.89 KMT2A (0.56) TSHRHSD17B10MEN1KMT2ANR1H2
SCHEMBL8939299 0.88 HDAC2 (0.47) TSHRHSD17B10HDAC2FDFT1
SCHEMBL9552934 0.87 MEN1 (0.43) TSHRHSD17B10MEN1KMT2AHIF1A
SCHEMBL9553047 0.86 TSHR (0.45) TSHRHSD17B10MEN1KMT2AHIF1A
SCHEMBL11744015 0.86 HDAC2 (0.49) TSHRHSD17B10HDAC2FDFT1
SCHEMBL9553611 0.84 MEN1 (0.44) TSHRHSD17B10MEN1KMT2ARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252252-A Longitudinal polarization MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1993-10-12 US disclosed
US-5120467-A Longitudinal polarization and-or cross-polarization MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-06-09 US disclosed
US-4723005-A CONTAINING POLARIZED CYANO OR HALOGEN SUBSTITUENTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1988-02-02 US disclosed
EP-0139996-A1 Anisotropic compounds and liquid crystal mixtures MERCK PATENT GmbH (DE) 1985-05-08 EP disclosed