SCHEMBL9564953

SCHEMBL9564953

O=S(=O)(c1nc2cncnc2n1Cc1ccc(F)cc1)C1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 19/20 0.54
CYP3A4 P08684 18/20 0.54
USP2 O75604 17/20 0.54
CYP2C19 P33261 14/20 0.54
ALDH1A1 P00352 11/20 0.54
LMNA P02545 6/20 0.54
TSHR P16473 5/20 0.54
CYP2C9 P11712 16/20 0.53
MAPK1 P28482 10/20 0.52
HIF1A Q16665 6/20 0.52
CYP2D6 P10635 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
HPGD P15428 3/20 0.49
ALOX15 P16050 1/20 0.49
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
CASP1 P29466 6/20 0.46
CASP7 P55210 6/20 0.46
HSD17B10 Q99714 5/20 0.44
TP53 P04637 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9564962 0.81 USP2 (0.50) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
SCHEMBL9539548 0.79 KCNH2 (0.61) CYP1A2CYP3A4CYP2C19CYP2C9CYP2D6
SCHEMBL9564851 0.78 CYP1A2 (0.54) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
SCHEMBL9565025 0.78 CYP1A2 (0.53) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
SCHEMBL9564845 0.78 KCNH2 (0.64) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
SCHEMBL9564917 0.78 CYP1A2 (0.53) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL9564856 0.77 KCNH2 (0.63) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
Oxalic Acid SCHEMBL9564888 0.76 CYP1A2 (0.51) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
Oxalic Acid SCHEMBL9564885 0.76 CYP1A2 (0.51) CYP1A2CYP3A4USP2CYP2C19ALDH1A1
Fumaric Acid SCHEMBL9876528 0.74 HRH1 (0.49) CYP1A2CYP3A4USP2CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed