SCHEMBL9565329

SCHEMBL9565329

Clc1ncc(-c2cccnc2)nc1C1CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.46
MAPK1 P28482 2/20 0.46
CYP3A4 P08684 3/20 0.43
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
HPGDS O60760 1/20 0.41
CYP19A1 P11511 3/20 0.41
ALDH1A1 P00352 4/20 0.40
CYP1A2 P05177 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
ACHE P22303 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PIM1 P11309 1/20 0.39
RECQL P46063 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565372 0.79 MAPK1 (0.49) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL9565316 0.76 CYP2A6 (0.43) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL9565318 0.72 PDGFRB (0.48) CYP2A6MAPK1CYP3A4HPGDSCYP19A1
SCHEMBL7424771 0.72 MAPK1 (0.48) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL7328164 0.70 CYP2A6 (0.45) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL7430012 0.69 CYP11B1 (0.50) CYP2A6MAPK1CYP3A4CYP19A1ALDH1A1
SCHEMBL7440831 0.69 CYP2A6 (0.44) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL7436678 0.68 CYP2A6 (0.43) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL24037028 0.67 CYP2A6 (0.52) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1
SCHEMBL30338445 0.67 CYP2A6 (0.52) CYP2A6MAPK1CYP3A4HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543245-A1 Renin inhibiting amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed
CN-1072413-A Amino acid derivative HOFFMANN LA ROCHE (CH) 1993-05-26 CN disclosed