SCHEMBL9569175

SCHEMBL9569175

CCOC(=O)Oc1cn2c3c(c(N4CCNC(C)C4)c(F)cc3c1=O)OC(C1CC1)=C2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 3/20 0.47
HSD17B10 Q99714 3/20 0.47
PMP22 Q01453 1/20 0.47
POLB P06746 1/20 0.45
PRKD3 O94806 1/20 0.45
ALOX15 P16050 1/20 0.45
OPRM1 P35372 1/20 0.45
CLK2 P49760 1/20 0.45
KCNH2 Q12809 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
TOP2A P11388 15/20 0.36
TOP2B Q02880 12/20 0.36
TOP1 P11387 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9569168 0.89 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9569148 0.83 STAT3 (0.38) KDM4EALDH1A1HPGDHSD17B10KCNH2
SCHEMBL9560219 0.81 KDM4E (0.51) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9560796 0.78 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10PMP22
Hydrochloric Acid SCHEMBL9569182 0.75 TOP2A (0.47) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL9560217 0.75 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9560446 0.74 KDM4E (0.52) KDM4EALDH1A1HPGDHSD17B10PMP22
Hydrochloric Acid SCHEMBL9560508 0.74 TOP1 (0.45) ALDH1A1POLBOPRM1TOP2ATOP2B
Hydrochloric Acid SCHEMBL9560156 0.73 TOP1 (0.46) TOP2ATOP2BTOP1
SCHEMBL9510219 0.72 KDM4E (0.51) KDM4EALDH1A1HPGDHSD17B10PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563734-A1 9-fluoro-7-oxo-7H-pyrido(1,2,3-de)(1,4)benzoxazine carboxylic acids and esters and their use as antiviral agents BAYER AG (DE) 1993-10-06 EP disclosed