SCHEMBL9570267

SCHEMBL9570267

NC(=O)c1ccc2nc(C[O])cn2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.46
AURKA O14965 1/20 0.46
DAPK3 O43293 1/20 0.46
JAK2 O60674 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PAK4 O96013 1/20 0.46
ABL1 P00519 1/20 0.46
NTRK1 P04629 1/20 0.46
FYN P06241 1/20 0.46
CSF1R P07333 1/20 0.46
RET P07949 1/20 0.46
MET P08581 1/20 0.46
PDGFRB P09619 1/20 0.46
PIM1 P11309 1/20 0.46
FGFR1 P11362 1/20 0.46
PDGFRA P16234 1/20 0.46
PRKACA P17612 1/20 0.46
FLT1 P17948 1/20 0.46
LTK P29376 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9597339 0.87 MCHR1 (0.50) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL10066171 0.86 CHEK1 (0.45) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL13384211 0.86 ABL1 (0.45) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL5401674 0.80 KDM4E (0.42) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL30845741 0.78 EGLN1 (0.52) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL29651927 0.78 KDM4E (0.43) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL10053505 0.77 MCHR1 (0.48) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL17336347 0.76 F7 (0.43) FYNRETGRK5CCNE1CDK2
SCHEMBL327269 0.75 PTGS1 (0.54) CHEK1AURKADAPK3JAK2PRKD3
SCHEMBL9570490 0.74 NPC1 (0.50) CDK5KDM4EALDH1A1POLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5270322-A Imidazo[1,2-a]pyridines, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1993-12-14 US disclosed
EP-0555825-A1 Imidazo(1,2-a)pyridines as angiotensin-II-antagonists Dr. Karl Thomae GmbH (DE) 1993-08-18 EP disclosed