SCHEMBL9574129

SCHEMBL9574129

BrCCCCCCOCCCCc1ccc2c(c1)OCO2

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.51
HDAC3 O15379 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
TAAR1 Q96RJ0 1/20 0.50
CALM1 P0DP23 2/20 0.49
HDAC8 Q9BY41 1/20 0.48
FAAH O00519 1/20 0.46
MGLL Q99685 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
MAOA P21397 1/20 0.45
MAOB P27338 1/20 0.45
HTR2A P28223 3/20 0.45
HTR2C P28335 3/20 0.45
HTR2B P41595 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070877 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL7564465 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL8077779 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL8063292 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL8077486 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL8062071 0.91 TAAR1 (0.59) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL8072554 0.89 TAAR1 (0.61) HDAC1HDAC3HDAC2HDAC6TAAR1
SCHEMBL11773030 0.87 CYP3A4 (0.49) TAAR1CALM1FAAHMGLL
SCHEMBL11773043 0.87 CYP3A4 (0.49) TAAR1CALM1FAAHMGLL
SCHEMBL11776870 0.87 CYP3A4 (0.49) TAAR1CALM1FAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5243076-A Adrenergic stimulant intermediates GLAXO GROUP LTD. 1993-09-07 US disclosed
US-5225445-A Respiratory system disorders GLAXO GROUP LTD. 1993-07-06 US disclosed
US-5126375-A Asthma, chronic bronchitis GLAXO GROUP LTD. (GB) 1992-06-30 US disclosed
US-5091422-A Treating inflammatory or allergic skin disease, lowering gastric acidity GLAXO GROUP LIMITED (GB) 1992-02-25 US disclosed
US-4992474-A Adrenergic stimulants GLAXO GROUP LTD. (GB) 1991-02-12 US disclosed