SCHEMBL9583202

SCHEMBL9583202

Nc1nc(NCc2ccc(OCc3ccccc3)cc2)nc2nc(-c3ccco3)nn12

nearest known ligand 0.81

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.81
ADORA3 P0DMS8 6/20 0.81
ADORA1 P30542 6/20 0.81
ADORA2B P29275 3/20 0.81
HDAC1 Q13547 9/20 0.69
HDAC6 Q9UBN7 7/20 0.69
ALDH1A1 P00352 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
CYP2C9 P11712 1/20 0.62
MAPK1 P28482 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.62
TMEM97 Q5BJF2 1/20 0.62
HSD17B10 Q99714 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834626 0.90 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL9325947 0.86 ADORA2A (0.77) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL9329053 0.85 ADORA2A (0.69) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL1754980 0.85 ADORA2A (0.83) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL29853688 0.85 ADORA2A (0.85) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL23928118 0.85 ADORA2A (0.73) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL9583900 0.85 ADORA2A (0.74) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL9429532 0.85 ADORA2A (0.60) ADORA2AADORA3ADORA1ADORA2BHDAC1
SCHEMBL9327402 0.83 ADORA2A (0.78) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL30676978 0.83 ADORA2A (0.69) ADORA2AADORA3ADORA1ADORA2BHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5246932-A Adenosine antagonist such as vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-09-21 US disclosed
EP-0515108-A2 Azolo (1,3,5) triazines as adenosine antagonists ZENECA LIMITED (GB) 1992-11-25 EP disclosed