SCHEMBL9583333

SCHEMBL9583333

CSc1nc(N)nc2c1ncn2COC(CO)CO

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 5/20 0.56
CYP3A4 P08684 4/20 0.56
ALDH1A1 P00352 2/20 0.56
MEN1 O00255 1/20 0.56
LMNA P02545 1/20 0.56
NFKB1 P19838 1/20 0.56
BLM P54132 1/20 0.56
VCP P55072 1/20 0.56
KMT2A Q03164 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
HK1 P19367 1/20 0.46
HKDC1 Q2TB90 1/20 0.46
SLC29A1 Q99808 3/20 0.46
PDE3A Q14432 1/20 0.45
CYP2C19 P33261 5/20 0.44
TDP1 Q9NUW8 1/20 0.42
CCNE1 P24864 4/20 0.41
CDK2 P24941 4/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10405081 0.88 HIF1A (0.54) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL9584901 0.86 PDE3A (0.49) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL9594486 0.83 PDE3A (0.48) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL9583894 0.83 BLM (0.48) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL9123481 0.83 BLM (0.62) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL10405077 0.82 HK1 (0.44) HIF1ACYP3A4ALDH1A1MEN1LMNA
Ganciclovir SCHEMBL14491348 0.82 BLM (0.60) HIF1ACYP3A4ALDH1A1MEN1LMNA
Ammonia Solution, Strong SCHEMBL10907047 0.82 BLM (0.60) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL9583704 0.81 MEN1 (0.57) HIF1ACYP3A4ALDH1A1MEN1LMNA
SCHEMBL11245765 0.81 PNP (0.56) HIF1ACYP3A4ALDH1A1MEN1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5250535-A Herpes virus; nontoxic; side effect reduction; humans and veterinary medicine SYNTEX INC. (US) 1993-10-05 US disclosed
US-4897479-A VIRICIDES FOR HERPES SIMPLEX MERCK & CO., INC. (US) 1990-01-30 US disclosed
US-4803271-A Process for preparing guanine derivatives SYNTEX (U.S.A.) INC. (US) 1989-02-07 US disclosed
EP-0105135-B1 SUBSTITUTED 9-(1-0- OR 3-0-MONOSUBSTITUTED OR 1,3-DI-0-SUBSTITUTED 1,3 DIHYDROXY-2-PROPOXYMETHYL) PURINES AS ANTIVIRAL AGENTS SYNTEX (U.S.A.) INC. (US) 1987-03-18 EP disclosed
US-4612314-A Substituted 9-(1 or 3-monoacyloxy or 1,3-diacyloxy-2-propoxymethyl) purines as antiviral agent SYNTEX (U.S.A.) INC. (US) 1986-09-16 US disclosed
US-4609661-A HERPES VIRUS SYNTEX (U.S.A.) INC. (US) 1986-09-02 US disclosed
US-4556659-A Substituted 9-(1-0- or 3-0-monosubstituted or 1,3-Di-0-substituted propoxymethyl)-purines as antiviral agents SYNTEX (U.S.A.) INC. (US) 1985-12-03 US disclosed
EP-0138683-A2 Purine derivatives, their application in anti-viral compositions MERCK & CO. INC. (US) 1985-04-24 EP disclosed
EP-0105135-A1 Substituted 9-(1-0- or 3-0-monosubstituted or 1,3-di-0-substituted 1,3 dihydroxy-2-propoxymethyl) purines as antiviral agents SYNTEX (U.S.A.) INC. (US) 1984-04-11 EP disclosed
EP-0085424-A2 Substituted 9-(1 or 3-monoacyloxy or 1,3-diacyloxy-2-propoxymethyl)purines as antiviral agent SYNTEX (U.S.A.) INC. (US) 1983-08-10 EP disclosed