SCHEMBL9587760

SCHEMBL9587760

O=C(O)c1ncsc1-c1cccc(I)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.69
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 1/20 0.44
THPO P40225 1/20 0.44
LMNA P02545 1/20 0.43
PMP22 Q01453 1/20 0.43
PDE4A P27815 1/20 0.37
HCRTR2 O43614 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
PTPN1 P18031 2/20 0.35
PTPRF P10586 1/20 0.35
PTPN2 P17706 1/20 0.35
HCRTR1 O43613 1/20 0.35
METAP2 P50579 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HKDC1 Q2TB90 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13398637 0.83 KDM4E (0.71) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL269667 0.82 KDM4E (1.00) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL1340272 0.82 KDM4E (0.69) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL985716 0.82 KDM4E (0.69) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL1338215 0.82 KDM4E (0.69) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL20376571 0.81 KDM4E (0.72) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL9588743 0.81 CYP1A2 (0.58) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL9586887 0.80 KDM4E (0.43) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL13398664 0.78 KDM4E (0.63) KDM4ECYP1A2CYP3A4THPOLMNA
SCHEMBL983442 0.78 KDM4E (0.63) KDM4ELMNAPTPN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5204482-A Ethylenediamine monoamide heteroaryl derivatives HOFFMAN-LAROCHE INC. (US) 1993-04-20 US disclosed
US-5011849-A Monoamine oxidase inhibitors HOFFMANN-LA ROCHE INC. (US) 1991-04-30 US disclosed