SCHEMBL9599549

SCHEMBL9599549

CC(C)c1cn2ccccc2c1S(=O)(=O)c1ccc(OCCCNCCc2ccccn2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HTR6 P50406 1/20 0.35
LMNA P02545 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC11 Q96DB2 2/20 0.34
HDAC8 Q9BY41 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9597712 0.87 MEN1 (0.45) RAB9ALMNACA12CA1CA2
SCHEMBL9599545 0.84 SCN8A (0.35) ALDH1A1TDP1HTTMEN1KMT2A
SCHEMBL9272756 0.84 MEN1 (0.43) ALDH1A1HTR6LMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL9599341 0.82 HRH3 (0.47) HTR6CA12CA1CA2CA9
SCHEMBL13940140 0.82 KMT2A (0.39) ALDH1A1CYP2C19CYP3A4HTR6LMNA
SCHEMBL4162892 0.82 MAPT (0.44) ALDH1A1CYP2C19CYP3A4HTR6LMNA
SCHEMBL8236467 0.81 POLB (0.39) ALDH1A1TDP1HTTCA12CA1
SCHEMBL6451740 0.80 MAPT (0.44) ALDH1A1CYP2C19CYP3A4HTR6LMNA
SCHEMBL4171578 0.80 HRH3 (0.37) RAB9AALDH1A1HTTCA12CA1
Hydrochloric Acid SCHEMBL9597718 0.79 SCN8A (0.40) ALDH1A1CYP3A4TDP1HTTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5182291-A Angina pectoris, hypotensive, antiarrhythmia, cerebral vascular insufficiency SANOFI (FR) 1993-01-26 US disclosed
US-5147878-A Hypotensive, antiarrhythmia agents SANOFI (FR) 1992-09-15 US disclosed
US-5039700-A Cardiovascular disorders, antitumor agents SANOFI (FR) 1991-08-13 US disclosed
US-5017579-A Use of aminoalkoxyphenyl derivatives for reducing and/or controlling excessive intraocular pressure SANOFI (FR) 1991-05-21 US disclosed
US-4957925-A HYPOTENSIVE AGENTS, ANTIARRHYTHMIA AGENTS, TREATMENT OF ANGINA SANOFI (FR) 1990-09-18 US disclosed