SCHEMBL9601879

SCHEMBL9601879

COC(=O)C1CC(CC(=O)O)CN1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.40
MMP2 P08253 3/20 0.38
ANPEP P15144 2/20 0.38
NR1H3 Q13133 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTPN1 P18031 1/20 0.38
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
P2RX3 P56373 1/20 0.35
HTRA1 Q92743 1/20 0.35
HSD17B10 Q99714 1/20 0.34
TGM2 P21980 1/20 0.34
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
ALDH1A1 P00352 1/20 0.33
UCHL1 P09936 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184330 1.00 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL19097280 1.00 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL17317642 1.00 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL29851070 0.89 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL6185885 0.89 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL31000687 0.89 NR1H2 (0.40) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL2708302 0.86 NR1H2 (0.51) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL18829250 0.86 NR1H2 (0.51) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL15815897 0.86 NR1H2 (0.41) NR1H2MMP2ANPEPNR1H3SMN1; SMN2
SCHEMBL2708360 0.86 NR1H2 (0.41) NR1H2MMP2ANPEPNR1H3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3152206-A1 ATX MODULATING AGENTS Biogen MA Inc. (US) 2017-04-12 EP disclosed
WO-2015188051-A1 ATX MODULATING AGENTS BIOGEN MA INC. (US) 2015-12-10 WO disclosed
US-5217963-A Antiischemic, antiepileptic agent CIBA-GEIGY CORPORATION (US) 1993-06-08 US disclosed
US-5057506-A Anticonvulsants, antispasmodic and antischemic agents CIBA-GEIGY CORPORATION (US) 1991-10-15 US disclosed
EP-0203891-B1 CERTAIN PHOSPHONIC ACIDS AND DERIVATIVES CIBA-GEIGY AG (CH) 1991-05-15 EP disclosed
US-4906621-A Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade CIBA-GEIGY CORPORATION (US) 1990-03-06 US disclosed
US-4898854-A NERVOUS SYSTEM DISORDERS CIBA-GEIGY CORPORATION (US) 1990-02-06 US disclosed
EP-0203891-A2 Certain phosphonic acids and derivatives CIBA-GEIGY AG (CH) 1986-12-03 EP disclosed