SCHEMBL9608842

SCHEMBL9608842

CCOC(=O)c1nc(COC)no1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
CACNA1F O60840 2/20 0.38
CACNA1D Q01668 2/20 0.38
CACNA1S Q13698 2/20 0.38
CACNA1C Q13936 2/20 0.38
CYP1A2 P05177 1/20 0.38
CHRM2 P08172 2/20 0.37
CHRM4 P08173 2/20 0.37
CHRM5 P08912 2/20 0.37
CHRM1 P11229 2/20 0.37
CHRM3 P20309 2/20 0.37
ALDH1A1 P00352 2/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA12 O43570 2/20 0.35
CA7 P43166 2/20 0.35
CA9 Q16790 2/20 0.35
CA14 Q9ULX7 2/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9461101 0.85 HTT (0.50) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL3559987 0.83 HTT (0.49) HTTCACNA1FCACNA1DCACNA1SCACNA1C
Hydrochloric Acid SCHEMBL3559985 0.82 HTT (0.48) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL2254343 0.82 HTT (0.48) HTTCACNA1FCACNA1DCACNA1SCACNA1C
Hydrochloric Acid SCHEMBL4493041 0.82 HTT (0.48) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL991667 0.81 HTT (0.47) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL1326830 0.80 CHRM2 (0.43) HTTCHRM2CHRM4CHRM5CHRM1
SCHEMBL15932331 0.79 HTT (0.46) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7400591 0.78 HTT (0.52) HTTCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL553588 0.75 KLKB1 (0.49) HTTCYP1A2ALDH1A1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069605-A1 NOVEL E,E-DIENE COMPOUNDS AND THEIR USE AS MEDICAMENTS AND COSMETICS DR. AUGUST WOLFF GMBH & CO. KG ARZNEIMITTEL (DE) 2012-05-31 WO disclosed