SCHEMBL9613192

SCHEMBL9613192

COC(=O)C1(NC(=O)c2ccc3c(C4CCCC4)cn(C)c3c2)CCC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 12/20 0.58
SCN5A Q14524 5/20 0.58
DGAT2 Q96PD7 1/20 0.43
CYP3A4 P08684 7/20 0.40
CYP2C19 P33261 7/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL899454 0.80 SCN9A (0.64) SCN9ASCN5ACYP3A4CYP2C19CYP2C9
SCHEMBL4972679 0.80 CYP3A4 (0.51) SCN9ADGAT2CYP3A4CYP2C19CYP1A2
SCHEMBL4975868 0.80 CYP3A4 (0.48) SCN9ADGAT2CYP3A4CYP2C19CYP1A2
SCHEMBL1260945 0.79 SCN9A (0.65) SCN9ASCN5ACYP3A4CYP2C19CYP2C9
SCHEMBL9613259 0.79 CYP3A4 (0.46) SCN9ADGAT2CYP3A4CYP2C19CYP1A2
SCHEMBL6367996 0.76 SCN9A (0.64) SCN9ASCN5A
SCHEMBL900323 0.76 SCN9A (0.64) SCN9ASCN5A
SCHEMBL4806227 0.74 CYP3A4 (0.69) SCN9ADGAT2CYP3A4CYP2C19CYP1A2
SCHEMBL12051156 0.73 SCN9A (0.51) SCN9ASCN5A
SCHEMBL899425 0.73 SCN9A (0.60) SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727797-B1 PROCESS FOR CROSS COUPLING INDOLES BOEHRINGER INGELHEIM PHARMA (US) 2012-05-30 EP disclosed
US-7332614-B2 Process for cross coupling indoles BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2008-02-19 US disclosed
US-7332614-B2 Process for cross coupling indoles BOEHRINGER INGELHEIM INTERNATIONAL, GMBH (DE) 2008-02-19 US disclosed