SCHEMBL9615152

SCHEMBL9615152

COc1ncc(C(F)(F)F)c(OC)n1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.49
KDR P35968 2/20 0.49
AURKB Q96GD4 2/20 0.49
CYP1A2 P05177 2/20 0.45
METAP2 P50579 1/20 0.45
CFTR P13569 3/20 0.37
QPCT Q16769 1/20 0.36
QPCTL Q9NXS2 1/20 0.36
ULK1 O75385 1/20 0.36
MAPK3 P27361 3/20 0.35
LRRK2 Q5S007 4/20 0.34
CRHR1 P34998 1/20 0.33
GAA P10253 1/20 0.33
CCR4 P51679 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9906411 0.84 GAA (0.39) AURKAKDRAURKBCYP1A2METAP2
SCHEMBL25526842 0.81 AURKA (0.49) AURKAKDRAURKBCFTRULK1
SCHEMBL15938761 0.79 AURKA (0.48) AURKAKDRAURKBCYP1A2METAP2
SCHEMBL3969157 0.79 XPO1 (0.38) AURKAKDRAURKBCYP1A2METAP2
SCHEMBL2015792 0.79 AURKA (0.48) AURKAKDRAURKBCYP1A2CFTR
SCHEMBL15938384 0.79 AURKA (0.50) AURKAKDRAURKBCYP1A2METAP2
SCHEMBL25199470 0.77 AURKA (0.49) AURKAKDRAURKBCFTRULK1
SCHEMBL31726555 0.77 AURKA (0.49) AURKAKDRAURKBCFTRULK1
SCHEMBL30397380 0.75 KDR (0.58) AURKAKDRAURKBCFTRULK1
SCHEMBL25207187 0.75 KDR (0.58) AURKAKDRAURKBCFTRULK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4117367-A None JP disclosed
JP-H04117367-A FLUOROALKYL GROUP-CONTAINING PYRIMIDINE DERIVATIVE AND PRODUCTION THEREOF AGENCY OF IND SCIENCE & TECHNOL 1992-04-17 JP disclosed