SCHEMBL9628356

SCHEMBL9628356

CN1[C@@H]2CC[C@H]1C[C@@H](Oc1nccc3ccccc13)C2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.52
SLC6A3 Q01959 2/20 0.52
CHRM2 P08172 4/20 0.47
CHRM5 P08912 4/20 0.47
CHRM1 P11229 4/20 0.47
CHRM3 P20309 4/20 0.47
CHRM4 P08173 3/20 0.47
HTR2C P28335 3/20 0.47
DRD2 P14416 2/20 0.47
DRD3 P35462 2/20 0.47
ADRA2C P18825 2/20 0.47
ADRA1D P25100 2/20 0.47
ADRA1A P35348 2/20 0.47
HRH1 P35367 2/20 0.47
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
DRD1 P21728 1/20 0.47
HRH2 P25021 1/20 0.47
HTR2A P28223 1/20 0.47
SLC6A4 P31645 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1178078 1.00 SLC6A2 (0.52) SLC6A2SLC6A3CHRM2CHRM5CHRM1
SCHEMBL1178075 1.00 SLC6A2 (0.52) SLC6A2SLC6A3CHRM2CHRM5CHRM1
Fumaric Acid SCHEMBL1177745 0.90 SLC6A2 (0.46) SLC6A2SLC6A3CHRM2CHRM5CHRM1
SCHEMBL1177925 0.79 SLC6A2 (0.59) SLC6A2SLC6A3CHRM2CHRM5CHRM1
SCHEMBL1177498 0.79 SLC6A2 (0.59) SLC6A2SLC6A3CHRM2CHRM5CHRM1
SCHEMBL5469724 0.74 ROCK1 (0.49) SLC6A2SLC6A3CHRM3HTR2CHRH1
Hydrochloric Acid SCHEMBL5476262 0.73 ROCK1 (0.48) SLC6A2CHRM3HTR2CHRH1HCRTR1
SCHEMBL29586291 0.73 HCRTR1 (0.47) HCRTR1HCRTR2MAPT
SCHEMBL21047726 0.73 HCRTR1 (0.47) HCRTR1HCRTR2MAPT
Hydrochloric Acid SCHEMBL29862550 0.73 ROCK1 (0.48) SLC6A2CHRM3HTR2CHRH1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082843-A PYRAZINYL AND PYRIDAZINYL ETHERS JOHN WYETH AND BROTHER LIMITED (GB) 1992-01-21 US disclosed
US-4929625-A Ethers JOHN WYETH AND BROTHERS LIMITED (GB) 1990-05-29 US disclosed