SCHEMBL9631503

SCHEMBL9631503

CCCCOc1ccc([C@H]2CC[C@H](CCC3CCC(CCC)CC3)CC2)c(F)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.37
CYP2C9 P11712 2/20 0.35
PPARG P37231 1/20 0.34
HTR1D P28221 2/20 0.34
HTR1B P28222 2/20 0.34
PTGES O14684 1/20 0.34
ALOX5 P09917 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRL1 P41146 4/20 0.33
HTR2C P28335 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9631507 1.00 SCN9A (0.37) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL4402652 0.99 SCN9A (0.38) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL26209537 0.99 SCN9A (0.38) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL9632575 0.96 SCN9A (0.34) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL9632579 0.96 SCN9A (0.34) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL9630413 0.95 CNR1 (0.35) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL14235296 0.95 SCN9A (0.36) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL9630415 0.95 CNR1 (0.35) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL26209558 0.95 SCN9A (0.36) SCN9ACYP2C9PPARGHTR1DHTR1B
SCHEMBL9631624 0.95 SCN9A (0.35) SCN9ACYP2C9PPARGHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0364538-B1 DIFLUOROBENZOL DERIVATIVES MERCK PATENT GmbH (DE) 1992-05-06 EP disclosed