SCHEMBL9636211

SCHEMBL9636211

CCOc1cc(OCC#N)ccc1-c1nc2cnccc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 7/20 0.40
CBFB Q13951 1/20 0.39
MELK Q14680 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PIP4K2A P48426 1/20 0.38
PDE3B Q13370 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9636094 0.96 CBFB (0.41) PDE5ACBFBKDM4ENPC1USP2
SCHEMBL9634527 0.94 PDE5A (0.39) PDE5ACBFBKDM4ENPC1ALDH1A1
SCHEMBL9636145 0.91 PDE5A (0.47) PDE5AMELKKDM4EALDH1A1LMNA
SCHEMBL7279872 0.90 CBFB (0.46) PDE5ACBFBKDM4ENPC1USP2
SCHEMBL9634582 0.90 PDE5A (0.40) PDE5ACBFBMELKKDM4ENPC1
SCHEMBL9635731 0.89 TOP1 (0.37) PDE5AKDM4EALDH1A1TP53PDE3B
SCHEMBL9634126 0.89 TOP1 (0.37) PDE5AKDM4EALDH1A1TP53PDE3B
SCHEMBL9636160 0.88 PDE2A (0.47) PDE5AKDM4ENPC1ALDH1A1HPGD
SCHEMBL9634827 0.88 PDE5A (0.41) PDE5AKDM4EALDH1A1HPGDPDE3B
SCHEMBL10740582 0.87 SMN1; SMN2 (0.40) PDE5ACBFBKDM4ENPC1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5104881-A 2-ARYLIMIDAZOPYRIDINES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-04-14 US disclosed
US-4616090-A 2-arylimidazopyridines intermediates MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1986-10-07 US disclosed