SCHEMBL9639591

SCHEMBL9639591

CCNc1cccnc1N1CCN(CCO)CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.50
CHIA Q9BZP6 1/20 0.46
METAP1 P53582 1/20 0.46
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 2/20 0.44
SIRT6 Q8N6T7 1/20 0.43
ACHE P22303 1/20 0.43
ELANE P08246 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
DRD4 P21917 1/20 0.42
HRH1 P35367 2/20 0.41
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 3/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9640177 0.99 PARP1 (0.49) PARP1CHIAMETAP1KDM4EALDH1A1
SCHEMBL9639730 0.92 PARP1 (0.48) PARP1CHIAMETAP1DRD4IDO1
Fumaric Acid SCHEMBL9755189 0.91 PARP1 (0.48) PARP1CHIAMETAP1KDM4EALDH1A1
Fumaric Acid SCHEMBL9639454 0.91 PARP1 (0.48) PARP1CHIAMETAP1KDM4EALDH1A1
SCHEMBL9689528 0.90 PARP1 (0.47) PARP1CHIADRD4
SCHEMBL9688155 0.90 PARP1 (0.47) PARP1CHIADRD4
SCHEMBL9689437 0.90 PARP1 (0.47) PARP1CHIADRD4
Hydrochloric Acid SCHEMBL9690356 0.89 PARP1 (0.46) PARP1CHIADRD4
Hydrochloric Acid SCHEMBL9690279 0.89 PARP1 (0.46) PARP1CHIADRD4
Hydrochloric Acid SCHEMBL9689424 0.89 PARP1 (0.46) PARP1CHIADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO claimed
EP-0496746-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1992-08-05 EP disclosed
WO-1991006542-A1 PHARMACEUTICALLY ACTIVE AMINO-SUBSTITUTED HETEROARYL AMINES THE UPJOHN COMPANY (US) 1991-05-16 WO disclosed