SCHEMBL9645681

SCHEMBL9645681

CC(C)Cc1ccc(C(C)(O)C(N)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.53
ALOX5 P09917 2/20 0.47
PTGS1 P23219 4/20 0.46
PTGS2 P35354 4/20 0.46
CXCR1 P25024 3/20 0.46
CXCR2 P25025 3/20 0.46
LMNA P02545 2/20 0.46
CYP2C9 P11712 2/20 0.46
AKR1C3 P42330 2/20 0.46
ALB P02768 1/20 0.46
ESR1 P03372 1/20 0.46
RARB P10826 1/20 0.46
ADRB3 P13945 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR2A P28223 1/20 0.46
NR1I3 Q14994 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
CXCL8 P10145 1/20 0.46
TSHR P16473 1/20 0.46
AKR1C2 P52895 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22722986 0.84 PTGS1 (0.51) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL7323204 0.84 PTGS1 (0.51) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL22722992 0.84 PTGS1 (0.51) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL11766801 0.84 PTGS1 (0.47) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL10749840 0.78 NR1H4 (0.46) ALOX5PTGS1PTGS2CXCR1CXCR2
SCHEMBL764935 0.77 PTGS1 (0.46) EPHX1ALOX5PTGS1PTGS2CXCR1
Dimethylamine SCHEMBL3820590 0.76 EPHX1 (0.46) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL30619574 0.76 PTGS1 (0.50) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL24473432 0.75 PTGS1 (0.47) EPHX1ALOX5PTGS1PTGS2CXCR1
SCHEMBL27901537 0.75 TSHR (0.51) EPHX1ALOX5PTGS1PTGS2CXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-57093923-A None JP disclosed
JP-52151144-A None JP disclosed
WO-2016069952-A1 ANTI-ACNE COMPOSITION AND METHODS OF USE RAYUDU SREEDHAR RAO (US) 2016-05-06 WO disclosed
US-5166434-A Process for the preparation of aromatic-substituted unsaturated amides ETHYL CORPORATION (US) 1992-11-24 US disclosed
JP-S5793923-A PREPARATION OF 2-(4-ISOBUTYLPHENYL) PROPIONIC ACID MITSUI TOATSU CHEM INC 1982-06-11 JP disclosed
JP-S52151144-A PREPARATION OF 2-SUBSTITUTED-ACRYLIC AMIDE AND 2-SUBSTITUTED-PROPIONIC ACID DERIVATIVES MITSUI TOATSU CHEM INC 1977-12-15 JP disclosed