SCHEMBL9651986

SCHEMBL9651986

Cc1cccc(C(=O)N(NC(=O)c2cccs2)C(C)(C)C)c1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 6/20 0.65
CYP3A4 P08684 2/20 0.56
CYP2C9 P11712 1/20 0.56
KCNK3 O14649 1/20 0.56
KCNK9 Q9NPC2 1/20 0.56
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
GAA P10253 1/20 0.53
PKM P14618 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
POLB P06746 1/20 0.50
ALDH1A1 P00352 1/20 0.47
MAPK1 P28482 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651981 0.90 ABCB1 (0.69) ABCB1CYP3A4CYP2C9KCNK3KCNK9
SCHEMBL9651949 0.86 NPC1 (0.58) ABCB1CYP3A4CYP2C9SMN1; SMN2POLB
SCHEMBL8172543 0.86 POLB (0.68) CYP3A4CYP2C9KMT2AMEN1SMN1; SMN2
SCHEMBL9714226 0.84 ABCB1 (0.89) ABCB1CYP3A4CYP2C9POLB
SCHEMBL9651153 0.82 MAPT (0.60) ABCB1CYP3A4CYP2C9KMT2AMEN1
SCHEMBL9507281 0.82 CYP3A4 (0.83) ABCB1CYP3A4CYP2C9POLB
SCHEMBL10722074 0.82 ABCB1 (0.89) ABCB1CYP3A4CYP2C9POLB
SCHEMBL9651116 0.81 ABCB1 (0.62) ABCB1CYP3A4CYP2C9POLB
SCHEMBL9714204 0.81 ABCB1 (0.78) ABCB1CYP3A4CYP2C9SMN1; SMN2POLB
SCHEMBL9652315 0.81 ABCB1 (0.69) ABCB1CYP3A4CYP2C9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0261755-B1 FIVE-MEMBERED HETEROCYCLIC DERIVATIVES OF N'-SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1992-12-16 EP disclosed