SCHEMBL9668491

SCHEMBL9668491

Cc1cc(CCCCCOc2cccc(C3=NCCO3)c2)on1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
BRD4 O60885 1/20 0.37
BRD2 P25440 1/20 0.37
CREBBP Q92793 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP19A1 P11511 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9668199 1.00 KCNH2 (0.38) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9666409 0.88 KCNH2 (0.50) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9668318 0.88 KCNH2 (0.50) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9705718 0.88 KCNH2 (0.50) KCNH2HRH3HDAC3HDAC4HDAC1
Disoxaril SCHEMBL147146 0.88 KCNH2 (0.50) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9666126 0.87 KCNH2 (0.51) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9862950 0.83 NPC1 (0.36) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9705703 0.83 SCARB1 (0.39) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9667787 0.83 SCARB1 (0.39) KCNH2HRH3HDAC3HDAC4HDAC1
SCHEMBL9668441 0.83 NPC1 (0.36) KCNH2HRH3HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0137242-B1 (SUBSTITUTED) PHENYL-ALIPHATIC-ISOXAZOLES USEFUL AS ANTIVIRAL AGENTS AND PREPARATION THEREOF STERLING WINTHROP INC. (US) 1992-05-13 EP disclosed
US-5002960-A Viricides for combating picornaviruses STERLING DRUG, INC. (US) 1991-03-26 US disclosed
US-4939267-A Viricides STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4843087-A OXAZOLINYL COMPOUNDS; RHINOVIRUSES AND PICORNAVIRUSES STERLING DRUG INC. (US) 1989-06-27 US disclosed
EP-0137242-A2 (Substituted) Phenyl-aliphatic-isoxazoles useful as antiviral agents and preparation thereof STERLING WINTHROP INC. (US) 1985-04-17 EP disclosed