SCHEMBL9670657

SCHEMBL9670657

COc1ccc(/C(=N/O)N2CCCc3cc(C4=NNC(=O)SC4C)ccc32)cc1OC

nearest known ligand 0.84

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.84
PDE3B Q13370 8/20 0.81
PDE3A Q14432 8/20 0.81
PDE4A P27815 13/20 0.42
PDE4B Q07343 13/20 0.42
PDE4C Q08493 13/20 0.42
PDE4D Q08499 13/20 0.42
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RORC P51449 1/20 0.37
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9670663 1.00 KCNH2 (0.84) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9671610 0.93 KCNH2 (0.73) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9671601 0.93 KCNH2 (0.73) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9639182 0.91 KCNH2 (0.81) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9639177 0.91 KCNH2 (0.81) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9639332 0.91 KCNH2 (1.00) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9638807 0.91 KCNH2 (0.81) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9638810 0.91 KCNH2 (0.81) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9639330 0.91 KCNH2 (1.00) KCNH2PDE3BPDE3APDE4APDE4B
SCHEMBL9639183 0.91 KCNH2 (0.80) KCNH2PDE3BPDE3APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0492257-A1 Thiadiazinone derivatives MERCK PATENT GmbH (DE) 1992-07-01 EP disclosed