SCHEMBL9670802

SCHEMBL9670802

COc1ccccc1OC1CCNC1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.63
HTR1A P08908 4/20 0.63
HTR2C P28335 6/20 0.56
HTR2B P41595 4/20 0.56
SLC6A3 Q01959 5/20 0.51
SLC6A4 P31645 4/20 0.51
PDE4B Q07343 1/20 0.51
HRH1 P35367 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8271827 1.00 SLC6A2 (0.63) SLC6A2HTR1AHTR2CHTR2BSLC6A3
SCHEMBL8271831 1.00 SLC6A2 (0.63) SLC6A2HTR1AHTR2CHTR2BSLC6A3
Hydrochloric Acid SCHEMBL4129951 0.98 SLC6A2 (0.61) SLC6A2HTR1AHTR2CHTR2BSLC6A3
Hydrochloric Acid SCHEMBL9132412 0.98 SLC6A2 (0.61) SLC6A2HTR1AHTR2CHTR2BSLC6A3
Hydrochloric Acid SCHEMBL4133478 0.98 SLC6A2 (0.61) SLC6A2HTR1AHTR2CHTR2BSLC6A3
SCHEMBL1780546 0.89 HRH1 (0.62) SLC6A2HTR1AHTR2CSLC6A3SLC6A4
Hydrochloric Acid SCHEMBL4100905 0.88 HRH1 (0.60) SLC6A2HTR1AHTR2CSLC6A3SLC6A4
SCHEMBL2297425 0.85 SLC6A2 (0.62) SLC6A2HTR1ASLC6A3SLC6A4
SCHEMBL3330561 0.83 HTR2C (0.67) SLC6A2HTR1AHTR2CHTR2BSLC6A3
SCHEMBL3175157 0.83 HTR2C (0.67) SLC6A2HTR1AHTR2CHTR2BSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1841758-B1 SUBSTITUTED TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LTD (GB) 2009-11-18 EP disclosed
EP-0338331-B1 1,3 DISUBSTITUTED PYRROLIDINES BAYER AG (DE) 1992-10-21 EP disclosed
EP-0338331-A1 1,3 Disubstituted Pyrrolidines BAYER AG (DE) 1989-10-25 EP disclosed
US-4377582-A HYPOTENSIVE AGENTS A. H. ROBINS COMPANY, INC. (US) 1983-03-22 US disclosed
US-4306065-A HYPOTENSIVE A. H. ROBINS COMPANY, INCORPORATED (US) 1981-12-15 US disclosed
US-RE28973-E PARKINSON'S DISEASE A. H. ROBINS COMPANY, INCORPORATED (US) 1976-09-21 US disclosed