SCHEMBL9677654

SCHEMBL9677654

CC(C)(C)N1CCOC(COc2ccccc2)C1.CC(C)(C)N1CCOC(c2cc(F)ccc2F)C1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 17/20 0.51
HRH3 Q9Y5N1 1/20 0.47
SIGMAR1 Q99720 1/20 0.46
EPHX2 P34913 1/20 0.44
PDK1 Q15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9641415 0.83 KDM1A (0.36)
SCHEMBL9641488 0.83 HRH3 (0.64) DRD4HRH3EPHX2PDK1
Hydrochloric Acid SCHEMBL9640901 0.82 HRH3 (0.62) DRD4HRH3EPHX2PDK1
Hydrochloric Acid SCHEMBL9640978 0.82 KDM1A (0.36)
SCHEMBL14208023 0.68 HRH3 (0.68) DRD4HRH3PDK1
SCHEMBL10747239 0.68 HTR2C (0.36) DRD4EPHX2
SCHEMBL1943731 0.68 DRD4 (0.44) DRD4HRH3EPHX2PDK1
SCHEMBL17166229 0.67 EPHX2 (0.52) DRD4HRH3EPHX2PDK1
SCHEMBL2296807 0.67 DRD3 (0.47)
SCHEMBL2295365 0.67 DRD3 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290122-B1 MORPHOLINE DERIVATIVES AND THEIR USE BEECHAM GROUP PLC (GB) 1992-12-23 EP claimed