SCHEMBL9688280

SCHEMBL9688280

COc1c(F)c(F)cc2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.50
HRH3 Q9Y5N1 1/20 0.50
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 5/20 0.49
GSK3B P49841 5/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 4/20 0.48
POLB P06746 1/20 0.48
PRKD3 O94806 1/20 0.48
ALOX15 P16050 1/20 0.48
OPRM1 P35372 1/20 0.48
CLK2 P49760 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TOP2A P11388 3/20 0.47
TOP2B Q02880 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PIK3CD O00329 1/20 0.47
PIK3R1 P27986 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508837 0.85 KCNH2 (0.64) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL30181127 0.85 KCNH2 (0.64) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL9501339 0.85 KCNH2 (0.55) KCNH2HRH3KDM4EALDH1A1GSK3B
Fluoride SCHEMBL5142968 0.83 KCNH2 (0.62) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL7495837 0.83 KCNH2 (0.51) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL5142970 0.82 KCNH2 (0.61) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL1344812 0.82 GSK3B (0.60) KCNH2HRH3KDM4EALDH1A1GSK3B
SCHEMBL5279361 0.82 KCNH2 (0.63) KCNH2HRH3KDM4EALDH1A1HPGD
SCHEMBL483223 0.81 KDM4E (0.65) KCNH2KDM4EALDH1A1GSK3BHPGD
SCHEMBL18467305 0.81 KCNH2 (0.43) KCNH2HRH3KDM4EALDH1A1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5097032-A Quinoline- and naphthyridine carboxylic acids, salts WARNER-LAMBERT COMPANY (US) 1992-03-17 US disclosed
EP-0265230-B1 SUBSTITUTED-6-FLUORO-4-OXO-1,4-DIHYDROQUINOLINE-3-CARBOXYLIC ACIDS, DERIVATIVES THEREOF, PHARMACEUTICAL COMPOSITIONS COMPRISING THE COMPOUNDS, AND PROCESSES FOR PRODUCING THE COMPOUNDS WARNER-LAMBERT COMPANY (US) 1992-01-08 EP disclosed
US-4822801-A 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-04-18 US disclosed