SCHEMBL9688792

SCHEMBL9688792

Clc1ccc2onc(Cn3ccnc3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.55
CYP11B1 P15538 5/20 0.51
CYP11B2 P19099 4/20 0.51
CYP2A6 P11509 1/20 0.51
CYP2B6 P20813 1/20 0.51
TBXAS1 P24557 4/20 0.51
CYP1A2 P05177 1/20 0.42
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
QPCT Q16769 1/20 0.42
CYP4Z1 Q86W10 1/20 0.42
QPCTL Q9NXS2 1/20 0.42
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9689124 0.88 CYP11B1 (0.55) CYP19A1CYP11B1CYP11B2CYP2A6CYP2B6
Hydrochloric Acid SCHEMBL9688636 0.83 MAPT (0.49) CYP19A1CYP11B1CYP11B2TBXAS1POLB
Hydrochloric Acid SCHEMBL9688615 0.83 CYP19A1 (0.50) CYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL9688409 0.83 CYP19A1 (0.54) CYP19A1CYP11B1CYP11B2TBXAS1ADRA2C
SCHEMBL9688353 0.80 CYP19A1 (0.52) CYP19A1CYP11B1CYP11B2TBXAS1CYP1A2
Hydrochloric Acid SCHEMBL9689248 0.80 CYP11B1 (0.53) CYP19A1CYP11B1CYP11B2TBXAS1CYP1A2
Hydrochloric Acid SCHEMBL9689549 0.77 CYP19A1 (0.51) CYP19A1CYP11B1CYP11B2TBXAS1CYP1A2
Hydrochloric Acid SCHEMBL9688740 0.77 KDM4E (0.54) CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL10570210 0.76 CYP19A1 (0.44) CYP19A1POLB
Hydrochloric Acid SCHEMBL9687814 0.75 MAPT (0.39) MAPTQPCTL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298921-B1 1,2-BENZISOXAZOLES AND 1,2-BENZISOTHIAZOLES CIBA-GEIGY AG (CH) 1992-12-23 EP disclosed
US-4957931-A ANTICONVULSANTS, TREATMENT OF EPILEPSY CIBA-GEIGY CORPORATION (US) 1990-09-18 US disclosed
US-4859691-A Certain 1,2-benzisoxazole derivatives CIBA-GEIGY CORPORATION (US) 1989-08-22 US disclosed
EP-0298921-A1 1,2-Benzisoxazoles and 1,2-benzisothiazoles CIBA-GEIGY AG (CH) 1989-01-11 EP disclosed