SCHEMBL9689181

SCHEMBL9689181

CC1(C)CC(N)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR3 O15455 1/20 0.45
AKR1B1 P15121 2/20 0.43
KDM1A O60341 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
AR P10275 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
TDP1 Q9NUW8 3/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HIF1A Q16665 1/20 0.37
TSHR P16473 2/20 0.37
MALT1 Q9UDY8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689179 1.00 TLR3 (0.45) TLR3AKR1B1KDM1ASIRT2CHRNB4
SCHEMBL621018 0.82 KDM1A (0.38) AKR1B1KDM1ACHRNB4CHRNA3NR3C1
SCHEMBL27280217 0.81 TLR3 (0.43) TLR3AKR1B1SIRT2CHRNB4CHRNA3
SCHEMBL7479500 0.77 HTR2C (0.42) AKR1B1SMN1; SMN2LMNAHTTTDP1
SCHEMBL8795599 0.77 AKR1B1 (0.44) TLR3AKR1B1SIRT2NR3C1SMN1; SMN2
SCHEMBL8795728 0.77 AKR1B1 (0.44) TLR3AKR1B1SIRT2ARSMN1; SMN2
SCHEMBL3409160 0.76 CNR1 (0.48) KDM1ASIRT2SMN1; SMN2MAPTLMNA
SCHEMBL3322619 0.76 TRPV1 (0.41) AKR1B1KDM1ACYP3A4
Hydrochloric Acid SCHEMBL6561142 0.76 HTR2C (0.41) AKR1B1SMN1; SMN2LMNAHTTTDP1
SCHEMBL6024931 0.76 TRPV1 (0.41) AKR1B1KDM1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5140031-A Pyranyl cyanoguanidine derivatives E. R. SQUIBB & SONS, INC. (US) 1992-08-18 US disclosed
EP-0401010-A2 Pyranyl cyanoguanidine derivatives E.R. Squibb & Sons, Inc. (US) 1990-12-05 EP disclosed