SCHEMBL9692152

SCHEMBL9692152

Clc1ccc(-c2nc3c(Cl)ccnc3[nH]2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 5/20 0.46
CDK1 P06493 5/20 0.46
CCNB1 P14635 5/20 0.46
CCNB3 Q8WWL7 5/20 0.46
GSK3A P49840 4/20 0.46
GSK3B P49841 4/20 0.46
CDK5 Q00535 2/20 0.46
CDK5R1 Q15078 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GAA P10253 2/20 0.45
MGAM O43451 1/20 0.45
SI P14410 1/20 0.45
MGAM2 Q2M2H8 1/20 0.45
MAPK13 O15264 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4148211 0.84 MGAM (0.57) CCNB2CDK1CCNB1CCNB3GSK3A
SCHEMBL17645693 0.83 AURKA (0.63) CCNB2CDK1CCNB1CCNB3GSK3A
SCHEMBL4909757 0.83 CCNB2 (0.43) CCNB2CDK1CCNB1CCNB3GSK3A
SCHEMBL4909647 0.82 KDM4E (0.47) CDK1GSK3AGSK3BCDK5KDM4E
SCHEMBL4907943 0.81 SCD (0.44) ALDH1A1SMN1; SMN2MAPK11MAPK14PARP1
SCHEMBL4148352 0.79 DHODH (0.49) MAPK14TNKSTNKS2PARP1
SCHEMBL4909019 0.79 RHEB (0.57) KDM4EALDH1A1NPC1PKMHPGD
SCHEMBL17290061 0.78 PARP1 (0.46) PARP1AURKA
SCHEMBL19418832 0.77 PRMT5 (0.61)
SCHEMBL15972401 0.77 PRMT5 (0.67)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255217-B1 FUSED IMIDAZOHETEROCYCLIC COMPOUNDS A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1992-01-22 EP disclosed
US-4948800-A MUSCLE RELAXANTS; ANTICONVULSANTS; ANXIOLYTIC AGENTS; 3-HYDROXYALKYL-PYRIDO(4,5-B OR-C)IMIDAZOLE COMPOUNDS A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-14 US disclosed
US-4914109-A ANTICONVULSANTS, ANTIANXIETY AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1990-04-03 US disclosed
US-4873251-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANTIANXIETY AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1989-10-10 US disclosed
US-4824951-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANXIOLYTIC AGENTS A. H. ROBINS COMPANY, INCORPORATED (US) 1989-04-25 US disclosed
US-4772600-A MUSCLE RELAXANTS, ANTICONVULSANTS, ANXIOLYTIC A. H. ROBINS COMPANY, INC. (US) 1988-09-20 US disclosed
EP-0255217-A1 Fused imidazoheterocyclic compounds A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1988-02-03 EP disclosed