SCHEMBL9696722

SCHEMBL9696722

CC(C)c1c(C#CCO[PH](=O)C[C@@H](O)CC(=O)O)c(-c2ccc(F)cc2)c2n1CCCC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 11/20 0.37
ABCB11 O95342 2/20 0.34
NR1I2 O75469 1/20 0.34
RHOC P08134 1/20 0.34
CYP3A4 P08684 1/20 0.34
THRB P10828 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
SLCO1B1 Q9Y6L6 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C9 P11712 3/20 0.32
TBXA2R P21731 2/20 0.32
ADRA1A P35348 2/20 0.32
ESR1 P03372 1/20 0.32
CHRM1 P11229 1/20 0.32
PDE4A P27815 1/20 0.32
ABCC3 O15438 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695389 1.00 HMGCR (0.37) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9696605 0.85 KMT2A (0.38) HMGCRKMT2A
SCHEMBL9696601 0.85 KMT2A (0.38) HMGCRKMT2A
SCHEMBL9696814 0.84
SCHEMBL9696808 0.84
SCHEMBL9696237 0.82 HMGCR (0.37) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9696231 0.82 HMGCR (0.37) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9696228 0.80 HMGCR (0.38) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9696239 0.80 HMGCR (0.38) HMGCRABCB11NR1I2RHOCCYP3A4
SCHEMBL9695383 0.80 HMGCR (0.37) HMGCRABCB11NR1I2RHOCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124453-A Treatment of corresponding aldehyde with lithium bis(tri-methylsilyl)amide E. R. SQUIBB & SONS, INC. (US) 1992-06-23 US disclosed
EP-0444532-A1 Phosphorus-containing HMG-CoA reductase inhibitors, new intermediates and method E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed
US-5025000-A Anticholesterol, antilipemic agents E. R. SQUIBB & SONS, INC. (US) 1991-06-18 US disclosed