SCHEMBL9699892

SCHEMBL9699892

CCc1cc(-n2cnc(C)c2)cc2c1NC(=O)SC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.35
PSEN1 P49768 5/20 0.35
PSEN2 P49810 5/20 0.35
APH1B Q8WW43 5/20 0.35
NCSTN Q92542 5/20 0.35
APH1A Q96BI3 5/20 0.35
PSENEN Q9NZ42 5/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NR2E1 Q9Y466 4/20 0.34
LDLR P01130 1/20 0.32
PCSK9 Q8NBP7 1/20 0.32
CYP2E1 P05181 1/20 0.32
CYP2A6 P11509 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700770 0.86 NR2E1 (0.36) CYP3A4PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL9701801 0.85 NR2E1 (0.35) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9700832 0.77 PSEN1 (0.46) CYP3A4PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL9701788 0.76 PSEN1 (0.45) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9700823 0.72 NR2E1 (0.36) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9700837 0.68 PDE3B (0.43) PDE4APDE4BPDE4CPDE4D
SCHEMBL9700769 0.66
SCHEMBL9699755 0.64 NR2E1 (0.36) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL9700879 0.64 PSEN1 (0.46) CYP3A4PSEN1PSEN2APH1BNCSTN
SCHEMBL22313383 0.62 CYP3A4 (0.49) CYP3A4PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0510235-A1 Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same DONG-A PHARM. CO., LTD. (KR) 1992-10-28 EP disclosed