SCHEMBL9702847

SCHEMBL9702847

Cc1sccc1-c1nc2cc3c(cc2[nH]1)C(C)(C)CC(=O)N3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
AURKA O14965 2/20 0.41
AURKB Q96GD4 2/20 0.41
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
ERAP1 Q9NZ08 1/20 0.35
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9380784 0.81 KDM4E (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9378391 0.80 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9383798 0.80 PDE3B (0.41) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9703439 0.79 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10699235 0.79 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9378253 0.78 PDE4A (0.54) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9702835 0.77 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9382509 0.77 PDE5A (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9379359 0.77 PDE3B (0.69) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9379360 0.77 AURKA (0.41) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed