SCHEMBL9708520

SCHEMBL9708520

Cn1c(=O)c2c(nc(C3CCCCC3)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(C)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.48
HSD17B10 Q99714 3/20 0.48
MAPK1 P28482 3/20 0.48
TP53 P04637 2/20 0.48
ADORA2A P29274 2/20 0.45
ADORA2B P29275 2/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
RECQL P46063 1/20 0.44
ALOX15 P16050 1/20 0.43
LMNA P02545 3/20 0.43
DPP4 P27487 2/20 0.43
MAPT P10636 1/20 0.43
AGTR1 P30556 2/20 0.43
AGTR2 P50052 2/20 0.43
HTT P42858 1/20 0.42
POLB P06746 1/20 0.41
BLM P54132 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708549 0.93 KMT2A (0.45) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9708135 0.93 KMT2A (0.43) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9707804 0.92 ADORA2A (0.46) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9707460 0.92 KMT2A (0.43) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9708269 0.92 ADORA2A (0.46) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9707343 0.91 KMT2A (0.44) TSHRHSD17B10MAPK1TP53KMT2A
SCHEMBL9707486 0.91 KMT2A (0.42) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9708066 0.91 KMT2A (0.44) TSHRHSD17B10MAPK1TP53KMT2A
SCHEMBL9707534 0.91 KMT2A (0.44) TSHRHSD17B10MAPK1TP53ADORA2A
SCHEMBL9707874 0.91 TRPC4 (0.43) TSHRHSD17B10MAPK1TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO claimed
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed