SCHEMBL9710101

SCHEMBL9710101

O=C1C[S+]([O-])c2ccccc2CN1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
AKR1C1 Q04828 1/20 0.33
AHR P35869 1/20 0.32
PDK2 Q15119 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PARP1 P09874 2/20 0.32
NPC1 O15118 1/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
PDPK1 O15530 1/20 0.31
PARP10 Q53GL7 1/20 0.31
PARP11 Q9NR21 1/20 0.31
TDP2 O95551 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9710113 0.77 PARP1 (0.37) PARP1PARP10TDP2
SCHEMBL17058245 0.74
SCHEMBL7385496 0.74
SCHEMBL9710333 0.73 SRD5A1 (0.33)
SCHEMBL9710530 0.73 PARP1 (0.37) PARP1PARP10PARP11
SCHEMBL88930 0.70 AHR (0.42) ALDH1A1AHRPDK2HSD17B10NPC1
SCHEMBL28606378 0.70 CA12 (0.35) CA12CA9AHRPDK2ALOX15
SCHEMBL28617213 0.70 CA12 (0.35) CA12CA9AHRPDK2ALOX15
SCHEMBL11560006 0.70 CA12 (0.35) CA12CA9AHRPDK2ALOX15
Hydrochloric Acid SCHEMBL20590674 0.69 CA12 (0.34) CA12CA9AHRPDK2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021668-A1 BENZOTHIAZEPINONES AND THEIR USE AS ANTICONVULSANTS THE BOOTS COMPANY PLC (GB) 1992-12-10 WO disclosed