SCHEMBL9710474

SCHEMBL9710474

N[C@@H](Cc1ccccc1)C(=O)C1NC(OC(=O)O)Cc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 5/20 0.42
ALPI P09923 1/20 0.41
PKM P14618 1/20 0.41
PTGS1 P23219 1/20 0.41
XIAP P98170 1/20 0.41
SLC7A5 Q01650 1/20 0.41
TYR P14679 1/20 0.38
SLC15A1 P46059 1/20 0.37
SLC1A3 P43003 2/20 0.36
SLC1A2 P43004 2/20 0.36
SLC1A1 P43005 2/20 0.36
LTA4H P09960 1/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11372279 0.87 TSHR (0.34)
SCHEMBL10698578 0.84 TSHR (0.37) XIAP
SCHEMBL9710472 0.83 HDAC8 (0.44) HDAC8ALPIPKMPTGS1XIAP
SCHEMBL10958377 0.78 ACE (0.46)
SCHEMBL2498951 0.77 HDAC8 (0.46) HDAC8SLC7A5
SCHEMBL10960540 0.77 IDO1 (0.36)
SCHEMBL10585437 0.75 XIAP (0.31) XIAP
SCHEMBL10604378 0.73 ACE (0.54)
SCHEMBL10589009 0.73 ACE (0.54)
SCHEMBL11051152 0.73 IDO1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016549-A1 PARASUBSTITUTED PHENYLALANINE DERIVATES PENTAPHARM AG (CH) 1992-10-01 WO disclosed