SCHEMBL9714835

SCHEMBL9714835

[CH2]COC(c1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.61
TDO2 P48775 4/20 0.61
IDO2 Q6ZQW0 2/20 0.61
SLC6A2 P23975 9/20 0.42
SLC6A4 P31645 9/20 0.42
SLC6A3 Q01959 9/20 0.42
KCNH2 Q12809 5/20 0.42
CYP3A4 P08684 5/20 0.42
CYP2D6 P10635 5/20 0.42
HTR1A P08908 2/20 0.40
HTR7 P34969 1/20 0.40
TNF P01375 1/20 0.39
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
SLC22A1 O15245 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9714864 0.98 IDO1 (0.64) IDO1TDO2IDO2SLC6A2SLC6A4
SCHEMBL1505811 0.82 SCN1A (0.50) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
Hydrochloric Acid SCHEMBL10654015 0.81 IDO1 (0.44) IDO1TDO2IDO2SLC6A2SLC6A4
SCHEMBL10577158 0.81 IDO1 (0.58) IDO1TDO2IDO2SLC6A2SLC6A4
SCHEMBL7429799 0.74 IDO1 (0.50) IDO1TDO2SLC6A2SLC6A4SLC6A3
SCHEMBL10571717 0.72 CYP1A2 (0.56) SLC6A2SLC6A4SLC6A3KCNH2CYP3A4
Hydrochloric Acid SCHEMBL9714844 0.72 IDO1 (0.54) IDO1TDO2SLC6A2SLC6A4SLC6A3
SCHEMBL16759094 0.69 IDO1 (0.55) IDO1TDO2IDO2SLC6A2SLC6A4
SCHEMBL17802363 0.68 SLC6A4 (0.54) IDO1TDO2IDO2SLC6A2SLC6A4
SCHEMBL2336595 0.68 IDO1 (0.51) IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116988-A Antiepileptic WARNER-LAMBERT CO. (US) 1992-05-26 US disclosed
US-5053521-A 3-amino butyric acid uptake inhibitors, antiepileptic agents WARNER-LAMBERT COMPANY (US) 1991-10-01 US disclosed
EP-0221572-B1 N-SUBSTITUTED 3-PIPERIDINE-OR 3-PYRIDINE-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF WARNER-LAMBERT COMPANY (US) 1991-09-25 EP disclosed
US-4910312-A Containing 1-(2-(bis((4-trifluoromethylphenyl)methoxy)-ethyl)-substitution WARNER-LAMBERT COMPANY (US) 1990-03-20 US disclosed
EP-0346927-A2 Various N-substituted 3-piperidine carboxylic acids or N-substituted 3-pyridine-carboxylic acids and derivatives thereof WARNER-LAMBERT COMPANY (US) 1989-12-20 EP disclosed
US-4772615-A ANTICONVULSANT FOR TREATING EPILEPSY WARNER-LAMBERT COMPANY (US) 1988-09-20 US disclosed
EP-0221572-A2 N-substituted 3-piperidine-or 3-pyridine-carboxylic acids and derivatives thereof WARNER-LAMBERT COMPANY (US) 1987-05-13 EP disclosed