SCHEMBL9717581

SCHEMBL9717581

C=CC(=O)c1ccc(OCC(=O)NCC(=O)O)c(Cl)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTA1 P08263 4/20 0.50
GSTP1 P09211 4/20 0.50
ALDH1A1 P00352 4/20 0.50
NPSR1 Q6W5P4 3/20 0.50
TSHR P16473 3/20 0.50
CYP2C9 P11712 2/20 0.50
TP53 P04637 2/20 0.50
LMNA P02545 2/20 0.50
MEN1 O00255 1/20 0.50
ABCC3 O15438 1/20 0.50
PLIN1 O60240 1/20 0.50
MAPT P10636 1/20 0.50
HSPD1 P10809 1/20 0.50
HTT P42858 1/20 0.50
RECQL P46063 1/20 0.50
MAP2K6 P52564 1/20 0.50
HSPE1 P61604 1/20 0.50
GSTO1 P78417 1/20 0.50
PLIN5 Q00G26 1/20 0.50
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9717604 0.88 CYP2C9 (0.62) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL9717560 0.81 GSTP1 (0.80) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL10833983 0.73 MAPT (0.58) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL10833252 0.73 MAPT (0.58) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL10833979 0.73 MAPT (0.58) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL11456708 0.73 CYP2C9 (0.64) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL27733269 0.71 TDP1 (0.74) ALDH1A1NPSR1TSHRTP53LMNA
SCHEMBL10834061 0.71 MAPT (0.59) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL10834067 0.71 MAPT (0.59) GSTA1GSTP1ALDH1A1NPSR1TSHR
SCHEMBL10834699 0.70 CYP2C9 (0.65) GSTA1GSTP1ALDH1A1NPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0240256-B1 COMPOUNDS USEFUL IN TREATING SICKLE CELL ANEMIA MERCK & CO. INC. (US) 1992-04-29 EP claimed
US-4699926-A Compounds useful in treating sickle cell anemia MERCK & CO., INC. (US) 1987-10-13 US claimed
EP-0240256-A2 Compounds useful in treating sickle cell anemia MERCK & CO. INC. (US) 1987-10-07 EP claimed
EP-0240256-B1 COMPOUNDS USEFUL IN TREATING SICKLE CELL ANEMIA MERCK & CO. INC. (US) 1992-04-29 EP disclosed
US-4699926-A Compounds useful in treating sickle cell anemia MERCK & CO., INC. (US) 1987-10-13 US disclosed
EP-0240256-A2 Compounds useful in treating sickle cell anemia MERCK & CO. INC. (US) 1987-10-07 EP disclosed